1-Alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: Development and Characterization of Adenosine A2B Receptor Antagonists and a New Radioligand with Subnanomolar Affinity and Subtype Specificity-Reference-Cited by-同舟云学术

1-Alkyl-8-(piperazine-1-sulfonyl)phenylxanthines: Development and Characterization of Adenosine A2B Receptor Antagonists and a New Radioligand with Subnanomolar Affinity and Subtype Specificity

Published:2009-05-27 Issue:13 Volume:52 Page:3994-4006
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Borrmann Thomas¹,Hinz Sonja¹,Bertarelli Daniela C. G.¹,Li Wenjin¹,Florin Nicole C.¹,Scheiff Anja B.¹,Müller Christa E.¹

Affiliation:

1. PharmaCenter Bonn, Pharmaceutical Institute, Pharmaceutical Chemistry I, An der Immenburg 4, D-53121 Bonn, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm900413e

Reference75 articles.

1. Airway effects of purine nucleosides and nucleotides and release with bronchial provocation in asthma

2. Adenosine in exhaled breath condensate in healthy volunteers and in patients with asthma

3. Adenosine in Bronchoalveolar Lavage Fluid in Asthma

4. Metabolic Consequences of Adenosine Deaminase Deficiency in Mice Are Associated with Defects in Alveogenesis, Pulmonary Inflammation, and Airway Obstruction

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