The Structural Basis for the Selectivity of Benzotriazole Inhibitors of PTP1B-Reference-Cited by-同舟云学术

The Structural Basis for the Selectivity of Benzotriazole Inhibitors of PTP1B

Published:2003-09-10 Issue:39 Volume:42 Page:11451-11459
ISSN:0006-2960
Container-title:Biochemistry
language:en
Short-container-title:Biochemistry

Author:

Scapin Giovanna¹,Patel Sangita B.¹,Becker Joseph W.¹,Wang Qingping¹,Desponts Caroline¹,Waddleton Deena¹,Skorey Kathryn¹,Cromlish Wanda¹,Bayly Christopher¹,Therien Michel¹,Gauthier Jacques Yves¹,Li Chun Sing¹,Lau Cheuk K.¹,Ramachandran Chidambaram¹,Kennedy Brian P.¹,Asante-Appiah Ernest¹

Affiliation:

1. Department of Medicinal Chemistry, Merck Research Laboratory, P. O. Box 2000, Rahway, New Jersey 07065, and Departments of Biochemistry & Molecular Biology and of Medicinal Chemistry, Merck Frosst Center for Therapeutic Research, P. O. Box 1005, Pointe-Claire - Dorval, Quebec, H9R 4P8, Canada

Publisher

American Chemical Society (ACS)

Subject

Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/bi035098j

Reference38 articles.

Cited by 108 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Regulation of protein phosphorylation by PTPN2 and its small-molecule inhibitors/degraders as a potential disease treatment strategy;European Journal of Medicinal Chemistry;2024-11

2. Elaborating azaaryl alkanes enabled by photoredox/palladium dual catalyzed dialkylation of azaaryl alkenes;Chinese Chemical Letters;2024-05

3. Discovery of PVD-06 as a Subtype-Selective and Efficient PTPN2 Degrader;Journal of Medicinal Chemistry;2023-11-15

4. Medicinal Aspects of PTP 1B Inhibitors as Anti-Breast Cancer Agents: An Overview;Current Medicinal Chemistry;2023-09-14

5. Identification of natural product inhibitors of PTP1B based on high-throughput virtual screening strategy: In silico, in vitro and in vivo studies;International Journal of Biological Macromolecules;2023-07