Selective Photoaffinity Probe That Enables Assessment of Cannabinoid CB2 Receptor Expression and Ligand Engagement in Human Cells-Reference-Cited by-同舟云学术

Selective Photoaffinity Probe That Enables Assessment of Cannabinoid CB2 Receptor Expression and Ligand Engagement in Human Cells

Published:2018-02-08 Issue:19 Volume:140 Page:6067-6075
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Soethoudt Marjolein^ORCID,Stolze Sara C.,Westphal Matthias V.¹,van Stralen Luuk²,Martella Andrea,van Rooden Eva J.,Guba Wolfgang³,Varga Zoltan V.⁴,Deng Hui^ORCID,van Kasteren Sander I.^ORCID,Grether Uwe³,IJzerman Adriaan P.^ORCID,Pacher Pal⁴,Carreira Erick M.¹,Overkleeft Herman S.,Ioan-Facsinay Andreea²,Heitman Laura H.,van der Stelt Mario

Affiliation:

1. Laboratorium für Organische Chemie, Eidgenössische Technische Hochschule Zürich, Vladimir-Prelog-Weg 3, Zürich 8093, Switzerland

2. Department of Rheumatology, Leiden University Medical Center, Albinusdreef 2, Leiden 2333 ZA, The Netherlands

3. Roche Innovation Center Basel, F. Hoffmann-La Roche Ltd., Grenzacherstrasse 124, Basel 4070, Switzerland

4. Laboratory of Cardiovascular Physiology and Tissue Injury, National Institute on Alcohol Abuse and Alcoholism, National Institutes of Health, 5625 Fishers Lane, Rockville, Maryland 20852, United States

Funder

Ministerie van Onderwijs, Cultuur en Wetenschap

Nederlandse Organisatie voor Wetenschappelijk Onderzoek

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

http://pubs.acs.org/doi/pdf/10.1021/jacs.7b11281

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