1. Laboratoire
de Chimie Organique, Institute of Chemistry, Biology and Innovation (CBI)-UMR 8231, ESPCI Paris, CNRS, PSL Research University, 10 rue Vauquelin 75231 Paris Cedex 05, France
2. Janssen Research & Development, Oncology Discovery Chemistry, Campus de Maigremont CS 10615, 27106 Cedex, Val de Reuil, France
3. Janssen Research & Development, Janssen Pharmaceutica NV Turnhoutseweg 30, 2340 Beerse, Belgium