Comparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines-Reference-Cited by-同舟云学术

Comparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines

Published:2017-03-08 Issue:6 Volume:82 Page:3239-3244
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Regenass Pierre¹,Bosc Damien¹,Riché Stéphanie¹,Gizzi Patrick²,Hibert Marcel¹,Karmazin Lydia³,Ganesan A.⁴,Bonnet Dominique¹^ORCID

Affiliation:

1. Laboratoire d’Innovation Thérapeutique, LabEx MEDALIS, Faculté de Pharmacie, UMR7200 CNRS/Université de Strasbourg, 74 route du Rhin, 67412 Illkirch, France

2. Université de Strasbourg, CNRS, Plateforme de Chimie Biologie Intégrative (PCBIS), UMS3286 and LabEx MEDALIS 6700 Strasbourg, France

3. Service de Cristallographie, Institut de Chimie de Strasbourg, BP 296/R8, 67008 Strasbourg, France

4. School of Pharmacy, University of East Anglia, Norwich Research Park, Norwich NR4 7TJ, U.K.

Funder

Université de Strasbourg

Centre National de la Recherche Scientifique

Labex MEDALIS

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.6b02895

Reference25 articles.

1. The rise, fall and reinvention of combinatorial chemistry

2. How were new medicines discovered?

3. Improvement in Aqueous Solubility in Small Molecule Drug Discovery Programs by Disruption of Molecular Planarity and Symmetry

4. Exploiting Chemical Diversity for Drug Discovery

5. A ring-distortion strategy to construct stereochemically complex and structurally diverse compounds from natural products

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