Application of Pd-Catalyzed Cross-Coupling Reactions in the Synthesis of 5,5-Dimethyl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazoles that Inhibit ALK5 Kinase-Reference-Cited by-同舟云学术

Application of Pd-Catalyzed Cross-Coupling Reactions in the Synthesis of 5,5-Dimethyl-5,6-dihydro-4H-pyrrolo[1,2-b]pyrazoles that Inhibit ALK5 Kinase

Published:2016-11-10 Issue:23 Volume:81 Page:11841-11856
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Tenora Lukáš¹,Galeta Juraj¹,Řezníčková Eva²,Kryštof Vladimír²,Potáček Milan¹

Affiliation:

1. Department of Chemistry, Faculty of Science, Masaryk University, Kotlářská 2, 611 37 Brno, Czech Republic

2. Laboratory of Growth Regulators, Faculty of Science, Palacký University & Institute of Experimental Botany ASCR, Šlechtitelů 27, 783 71 Olomouc, Czech Republic

Funder

Grantová Agentura Ceské Republiky

Univerzita Palackého v Olomouci

Central European Institute of Technology

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.joc.6b02230

Reference46 articles.

1. Palladium-Catalyzed Deaminative Phenanthridinone Synthesis from Aniline via C–H Bond Activation

2. Pd-Catalyzed sequential β-C(sp3)–H arylation and intramolecular amination of δ-C(sp2)–H bonds for synthesis of quinolinones via an N,O-bidentate directing group

3. Palladium-catalysed transannular C–H functionalization of alicyclic amines

4. Mild metal-catalyzed C–H activation: examples and concepts

5. Metal-free catalytic C-H bond activation and borylation of heteroarenes

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