Pyrazole Ligands: Structure−Affinity/Activity Relationships and Estrogen Receptor-α-Selective Agonists-Reference-Cited by-同舟云学术

Pyrazole Ligands: Structure−Affinity/Activity Relationships and Estrogen Receptor-α-Selective Agonists

Published:2000-11-28 Issue:26 Volume:43 Page:4934-4947
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Stauffer Shaun R.¹,Coletta Christopher J.¹,Tedesco Rosanna¹,Nishiguchi Gisele¹,Carlson Kathryn¹,Sun Jun¹,Katzenellenbogen Benita S.¹,Katzenellenbogen John A.¹

Affiliation:

1. Departments of Chemistry, Physiology, and Cell and Structural Biology, University of Illinois and University of Illinois College of Medicine, Urbana, Illinois 61801

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm000170m

Reference32 articles.

1. The estradiol pharmacophore: Ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding site

2. Molecular basis of agonism and antagonism in the oestrogen receptor

3. Different Residues of the Human Estrogen Receptor Are Involved in the Recognition of Structurally Diverse Estrogens and Antiestrogens

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