Design and Synthesis of a Potent and Selective Peptidomimetic Inhibitor of Caspase-3-Reference-Cited by-同舟云学术

Design and Synthesis of a Potent and Selective Peptidomimetic Inhibitor of Caspase-3

Published:2004-11-18 Issue:26 Volume:47 Page:6455-6458
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Micale Nicola¹,Vairagoundar Rajendran¹,Yakovlev Alexander G.¹,Kozikowski Alan P.¹

Affiliation:

1. Department of Medicinal Chemistry and Pharmacognosy, University of Illinois at Chicago, 833 South Wood Street, Illinois 60612, ChemBridge Research Laboratories, 16981 Via Tazon, San Diego, California 92127, and Georgetown University Medical Center, 3970 Reservoir Road, Washington, D.C. 20057

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm049248f

Reference32 articles.

1. From bench to clinic with apoptosis-based therapeutic agents

2. A novel heterodimeric cysteine protease is required for interleukin-1βprocessing in monocytes

3. The C. elegans cell death gene ced-3 encodes a protein similar to mammalian interleukin-1β-converting enzyme

4. Inactivation of Interleukin-1.beta. Converting Enzyme by Peptide (Acyloxy)methyl Ketones

5. Caspases: Intracellular Signaling by Proteolysis

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