Pilot Plant Preparation of tert-Butyl-4-(2-hydroxyethyl)-4-(pyrrolidin-1-yl)-piperidine-1-carboxylate, An Intermediate of Novel Antiarteriosclerotics, Via a Safe, Scalable Reformatsky-Type Reaction-Reference-Cited by-同舟云学术

Pilot Plant Preparation of tert-Butyl-4-(2-hydroxyethyl)-4-(pyrrolidin-1-yl)-piperidine-1-carboxylate, An Intermediate of Novel Antiarteriosclerotics, Via a Safe, Scalable Reformatsky-Type Reaction

Published:2011-08-15 Issue:6 Volume:15 Page:1433-1437
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Osato Hiroshi¹,Osaki Motonari¹,Oyama Takao¹,Takagi Youhei¹,Hida Takemasa¹,Nishi Koichi¹,Kabaki Mikio¹

Affiliation:

1. Chemical Development Center, CMC Development Laboratories, Shionogi & Co., Ltd., 1-3, Kuise Terajima 2-Chome, Amagasaki, Hyogo 660-0813, Japan

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op2001723

Reference21 articles.

1. Neue Synthese zweiatomiger einbasischer Säuren aus den Ketonen

2. Preparation and reactions of polyfunctional organozinc reagents in organic synthesis

3. The Reformatsky reaction in organic synthesis. Recent advances

4. Reformatsky Reactions Meet Catalysis and Stereoselectivity

5. Chemical reaction engineering for safety

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