Development of a Selective Peptide Macrocycle Inhibitor of Coagulation Factor XII toward the Generation of a Safe Antithrombotic Therapy-Reference-Cited by-同舟云学术

Development of a Selective Peptide Macrocycle Inhibitor of Coagulation Factor XII toward the Generation of a Safe Antithrombotic Therapy

Published:2013-04-25 Issue:9 Volume:56 Page:3742-3746
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Baeriswyl Vanessa¹,Calzavarini Sara²,Gerschheimer Christiane²,Diderich Philippe¹,Angelillo-Scherrer Anne²,Heinis Christian¹

Affiliation:

1. Institute of Chemical Sciences and Engineering, Ecole Polytechnique Fédérale de Lausanne (EPFL), CH-1015 Lausanne, Switzerland

2. Service and Central Laboratory of Hematology, Lausanne University Hospital, Rue du Bugnon 46, CH-1011 Lausanne, Switzerland

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm400236j

Reference25 articles.

1. Defective thrombus formation in mice lacking coagulation factor XII

2. Factor XI and XII as antithrombotic targets

3. Coleman, R. W.Contact Activation (Kallikrein–Kinnin) Pathway: Multiple Physiologic and Pathophysiologic Activities,5th ed;Lippincott Williams & Wilkins:Philadelphia, PA, 2006; pp107–130.

4. Ir-CPI, a coagulation contact phase inhibitor from the tick Ixodes ricinus, inhibits thrombus formation without impairing hemostasis

5. Factor XIIa Inhibitor Recombinant Human Albumin Infestin-4 Abolishes Occlusive Arterial Thrombus Formation Without Affecting Bleeding

Cited by 57 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Steps Toward Recapitulating Endothelium: A Perspective on the Next Generation of Hemocompatible Coatings;Macromolecular Bioscience;2024-07-29

2. Diversification of Phage-Displayed Peptide Libraries with Noncanonical Amino Acid Mutagenesis and Chemical Modification;Chemical Reviews;2024-04-30

3. Supercomputer Search for Coagulation Factor XIIa Inhibitors in the Chinese National Compound Library;Lecture Notes in Computer Science;2023

4. Experimentally Validated Novel Factor XIIa Inhibitors Identified by Docking and Quantum Chemical Post‐processing;Molecular Informatics;2022-11-21

5. MOrPH-PhD: A System for the Functional Selection of Genetically Encoded;Methods in Molecular Biology;2021-10-02