Asymmetric Synthesis of Telcagepant, a CGRP Receptor Antagonist for the Treatment of Migraine-Reference-Cited by-同舟云学术

Asymmetric Synthesis of Telcagepant, a CGRP Receptor Antagonist for the Treatment of Migraine

Published:2010-10-18 Issue:22 Volume:75 Page:7829-7841
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Xu Feng¹,Zacuto Michael¹,Yoshikawa Naoki¹,Desmond Richard¹,Hoerrner Scott¹,Itoh Tetsuji¹,Journet Michel¹,Humphrey Guy R.¹,Cowden Cameron¹,Strotman Neil¹,Devine Paul¹

Affiliation:

1. Department of Process Research, Merck Research Laboratories, Rahway, New Jersey 07065, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo101704b

Reference55 articles.

1. Migraine — Current Understanding and Treatment

2. The Global Burden of Headache: A Documentation of Headache Prevalence and Disability Worldwide

3. Calcitonin Gene-Related Peptide (CGRP) and Migraine

4. Calcitonin Gene-Related Peptide Antagonists as Treatments of Migraine and Other Primary Headaches

5. Blockade of CGRP Receptors in the Intracranial Vasculature: A New Target in the Treatment of Headache

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