Structure-Based Design of PDZ Ligands as Inhibitors of 5-HT2A Receptor/PSD-95 PDZ1 Domain Interaction Possessing Anti-hyperalgesic Activity-Reference-Cited by-同舟云学术

Structure-Based Design of PDZ Ligands as Inhibitors of 5-HT2A Receptor/PSD-95 PDZ1 Domain Interaction Possessing Anti-hyperalgesic Activity

Published:2013-08-23 Issue:10 Volume:8 Page:2209-2216
ISSN:1554-8929
Container-title:ACS Chemical Biology
language:en
Short-container-title:ACS Chem. Biol.

Author:

Vogrig Alexandre¹²,Dorr Liam³,Bouzidi Naoual¹²,Boucherle Benjamin¹²,Wattiez Anne-Sophie⁴⁵,Cassier Elisabeth⁶,Vallon Gary²⁷,Ripoche Isabelle²⁷,Abrunhosa-Thomas Isabelle²⁷,Marin Philippe⁶,Nauton Lionel¹²,Thery Vincent¹²,Courteix Christine⁴⁵,Lian Lu-Yun³,Ducki Sylvie²⁷

Affiliation:

1. Clermont Université, Université Blaise Pascal, Institut de Chimie de Clermont-Ferrand, BP 10448, F-63000 Clermont-Ferrand, France

2. CNRS, UMR6296, ICCF, F-63171 Aubiere, France

3. NMR Centre for Structural Biology, University of Liverpool, L6972B Liverpool, U.K.

4. Clermont Université, Université d’Auvergne, Pharmacologie Fondamentale et Clinique de la Douleur, BP 10448, F-63000 Clermont-Ferrand, France

5. Inserm, UMR1107, Neuro-Dol, F-63001 Clermont-Ferrand, France

6. Institut de Génomique Fonctionalle, CNRS UMR5203 − INSERM U661, Universités Montpellier 1&2, F-34094 Montpellier, France

7. Clermont Université, ENSCCF, Institut de Chimie de Clermont-Ferrand, BP 10448, F-63000 Clermont-Ferrand, France

Publisher

American Chemical Society (ACS)

Subject

Molecular Medicine,General Medicine,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/cb400308u

Reference31 articles.

1. Recognition of Unique Carboxyl-Terminal Motifs by Distinct PDZ Domains

2. PDZ domains in synapse assembly and signalling

3. Plasticity of PDZ domains in ligand recognition and signaling

Cited by 16 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Evolution of Artificial Arginine Analogues—Fluorescent Guanidiniocarbonyl-Indoles as Efficient Oxo-Anion Binders;Molecules;2022-05-07

2. Rational Design of PDZ Domain Inhibitors: Discovery of Small Organic Compounds Targeting PDZ Domains;Methods in Molecular Biology;2021

3. International Union of Basic and Clinical Pharmacology. CX. Classification of Receptors for 5-hydroxytryptamine; Pharmacology and Function;Pharmacological Reviews;2020-12-22

4. The serotonin receptor 2A (HTR2A) rs6313 variant is associated with higher ongoing pain and signs of central sensitization in neuropathic pain patients;European Journal of Pain;2020-12-03

5. Synthesis and biological activities of new pyrrolocarbazole-imidazobenzimidazole conjugates;Tetrahedron Letters;2020-07