4-Aryl-5-(4-Piperidyl)-3-Isoxazolol GABAA Antagonists: Synthesis, Pharmacology, and Structure−Activity Relationships-Reference-Cited by-同舟云学术

4-Aryl-5-(4-Piperidyl)-3-Isoxazolol GABAA Antagonists: Synthesis, Pharmacology, and Structure−Activity Relationships

Published:2007-03-22 Issue:8 Volume:50 Page:1988-1992
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Frølund Bente¹,Jensen Lars S.¹,Storustovu Signe I.¹,Stensbøl Tine B.¹,Ebert Bjarke¹,Kehler Jan¹,Krogsgaard-Larsen Povl¹,Liljefors Tommy¹

Affiliation:

1. Department of Medicinal Chemistry, Faculty of Pharmaceutical Sciences, University of Copenhagen, DK-2100 Copenhagen, Denmark, and Department of Molecular Pharmacology, Electrophysiology, and Medicinal Chemistry, H. Lundbeck A/S, DK-2500 Valby, Denmark

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm070038n

Reference16 articles.

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2. A new class of GABA agonist

3. GABA-A Receptor Ligands and their Therapeutic Potentials

4. Which GABAA-receptor subtypes really occur in the brain?

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