2-Phenyl-4-quinolinecarboxamides: A Novel Class of Potent and Selective Non-Peptide Competitive Antagonists for the Human Neurokinin-3 Receptor-Reference-Cited by-同舟云学术

2-Phenyl-4-quinolinecarboxamides: A Novel Class of Potent and Selective Non-Peptide Competitive Antagonists for the Human Neurokinin-3 Receptor

Published:1996-01-01 Issue:12 Volume:39 Page:2281-2284
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Giardina Giuseppe A. M.¹,Sarau Henry M.¹,Farina Carlo¹,Medhurst Andrew D.¹,Grugni Mario¹,Foley James J.¹,Raveglia Luca F.¹,Schmidt Dulcie B.¹,Rigolio Roberto¹,Vassallo Marco¹,Vecchietti Vittorio¹,Hay Douglas W. P.¹

Affiliation:

1. Department of Chemistry, SmithKline Beecham S.p.A., Via Zambeletti, 20021 Baranzate, Milano, Italy, Department of Pulmonary Pharmacology, SmithKline Beecham Pharmaceuticals, 709 Swedeland Road, King of Prussia, Pennsylvania 19406-0939, and Department of Neurology Research, SmithKline Beecham Pharmaceuticals, New Frontiers Science Park, Third Avenue, Harlow, Essex, England CM19 5AW

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm9602423

Reference28 articles.

1. Tachykinins

2. New selective agonists for neurokinin receptors: pharmacological tools for receptor characterization

3. Tachykinin receptors and tachykinin receptor antagonists

4. Mammalian Tachykinin Receptors

5. A Potent Nonpeptide Antagonist of the Substance P (NK 1 ) Receptor

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