Drug-to-Genome-to-Drug, Step 2: Reversing Selectivity in a Series of Antiplasmodial Compounds-Reference-Cited by-同舟云学术

Drug-to-Genome-to-Drug, Step 2: Reversing Selectivity in a Series of Antiplasmodial Compounds

Published:2012-01-24 Issue:3 Volume:55 Page:1274-1286
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Beghyn Terence B.¹²³⁴,Charton Julie¹²³⁴,Leroux Florence¹²³⁴,Henninot Antoine¹²³⁴,Reboule Irena¹²³⁴,Cos Paul⁵,Maes Louis⁵,Deprez Benoit¹²³⁴

Affiliation:

1. INSERM U761 Biostructures and Drug Discovery, Lille F-59006, France

2. Faculté de Pharmacie, Université Lille 2, Lille F-59006, France

3. Institut Pasteur de Lille, Lille F-59021, France

4. PRIM (), Lille, France

5. Laboratory of Microbiology, Parasitology, and Hygiene (LMPH), Faculty of Pharmaceutical, Biomedical, and Veterinary Sciences, University of Antwerp, B-2020 Antwerp, Belgium

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm201422e

Reference21 articles.

1. Drug to Genome to Drug: Discovery of New Antiplasmodial Compounds

2. Design, synthesis and biological activity of β-carboline-based type-5 phosphodiesterase inhibitors

3. Synthesis of Commercial Phosphodiesterase(V) Inhibitors

4. Structural Basis for the Activity of Drugs that Inhibit Phosphodiesterases

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