Orally Active Fumagillin Analogues: Transformations of a Reactive Warhead in the Gastric Environment-Reference-Cited by-同舟云学术

Orally Active Fumagillin Analogues: Transformations of a Reactive Warhead in the Gastric Environment

Published:2013-03-04 Issue:4 Volume:4 Page:381-386
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Arico-Muendel Christopher C.¹,Blanchette Heather¹,Benjamin Dennis R.¹,Caiazzo Teresa M.¹,Centrella Paolo A.¹,DeLorey Jennifer¹,Doyle Elisabeth G.¹,Johnson Steven R.¹,Labenski Matthew T.¹,Morgan Barry A.¹,O’Donovan Gary¹,Sarjeant Amy A.¹,Skinner Steven¹,Thompson Charles D.¹,Griffin Sarah T.¹,Westlin William¹,White Kerry F.¹

Affiliation:

1. Praecis Pharmaceuticals, Inc., 830 Winter Street, Waltham, Massachusetts 02451-1420, United States, and Department of Chemistry, Northwestern University, 2145 Sheridan Road, Evanston, Illinois 60208, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ml3003633

Reference24 articles.

1. The resurgence of covalent drugs

2. Covalent Modifiers: An Orthogonal Approach to Drug Design

3. Molecular recognition of angiogenesis inhibitors fumagillin and ovalicin by methionine aminopeptidase 2

4. Structure of Human Methionine Aminopeptidase-2 Complexed with Fumagillin

5. Fumagalone, a Reversible Inhibitor of Type 2 Methionine Aminopeptidase and Angiogenesis

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