Large-Scale Preparation of 2-Methyloxazole-4-carboxaldehyde-Reference-Cited by-同舟云学术

Large-Scale Preparation of 2-Methyloxazole-4-carboxaldehyde

Published:2007-11-20 Issue:1 Volume:12 Page:88-95
ISSN:1083-6160
Container-title:Organic Process Research & Development
language:en
Short-container-title:Org. Process Res. Dev.

Author:

Benoit Georges-Emmanuel¹,Carey John S.¹,Chapman Alan M.¹,Chima Ranjit¹,Hussain Nigel¹,Popkin Matthew E.¹,Roux Guillaume¹,Tavassoli Bahareh¹,Vaxelaire Carine¹,Webb Michael R.¹,Whatrup David¹

Affiliation:

1. Synthetic Chemistry, GlaxoSmithKline Pharmaceuticals, Old Powder Mills, Leigh, nr. Tonbridge, Kent TN11 9AN, U.K.

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/op700198s

Reference47 articles.

1. Analysis of the reactions used for the preparation of drug candidate molecules

2. References for the preparation of oxazole aldehyde1where experimental details are provided:

3. Synthesis of 4-Arylethynyl-2-methyloxazole Derivatives as mGluR5 Antagonists for Use in the Treatment of Drug Abuse

4. Synthesis and Structure−Activity Relationships of 3-[(2-Methyl-1,3-thiazol-4-yl)ethynyl]pyridine Analogues as Potent, Noncompetitive Metabotropic Glutamate Receptor Subtype 5 Antagonists; Search for Cocaine Medications

5. Enantioselective Total Synthesis of the Antitumor Macrolide Rhizoxin D

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