Fragment-Sized Thiazoles in Fragment-Based Drug Discovery Campaigns: Friend or Foe?-Reference-Cited by-同舟云学术

Fragment-Sized Thiazoles in Fragment-Based Drug Discovery Campaigns: Friend or Foe?

Published:2022-11-03 Issue:12 Volume:13 Page:1905-1910
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Proj Matic¹^ORCID,Hrast Martina¹^ORCID,Knez Damijan¹^ORCID,Bozovičar Krištof¹,Grabrijan Katarina¹,Meden Anže¹^ORCID,Gobec Stanislav¹^ORCID,Frlan Rok¹^ORCID

Affiliation:

1. Faculty of Pharmacy, University of Ljubljana, Askerceva 7, Ljubljana 1000, Slovenia

Funder

Javna Agencija za Raziskovalno Dejavnost RS

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.2c00429

Reference37 articles.

1. Thiazoles, Their Benzofused Systems, and Thiazolidinone Derivatives: Versatile and Promising Tools to Combat Antibiotic Resistance

2. 11. Thiazole: A privileged scaffold in drug discovery

3. Thiazoles: having diverse biological activities

4. Fragment-Based Screening of the Bromodomain of ATAD2

5. Discovery of small-molecule inhibitors targeting the ribosomal peptidyl transferase center (PTC) of M. tuberculosis

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