Discovery of 5-Phenyl-N-(pyridin-2-ylmethyl)-2-(pyrimidin-5-yl)quinazolin-4-amine as a Potent IKur Inhibitor-Reference-Cited by-同舟云学术

Discovery of 5-Phenyl-N-(pyridin-2-ylmethyl)-2-(pyrimidin-5-yl)quinazolin-4-amine as a Potent IKur Inhibitor

Published:2016-07-05 Issue:9 Volume:7 Page:831-834
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Finlay Heather J.¹²,Johnson James A.¹²,Lloyd John L.¹²,Jiang Ji¹²,Neels James¹²,Gunaga Prashantha¹²,Banerjee Abhisek¹²,Dhondi Naveen¹²,Chimalakonda Anjaneya¹²,Mandlekar Sandhya¹²,Conder Mary Lee¹²,Sale Harinath¹²,Xing Dezhi¹²,Levesque Paul¹²,Wexler Ruth R.¹²

Affiliation:

1. Departments of Discovery Chemistry, ‡Biology, and §Preclinical Candidate Optimization, Bristol-Myers Squibb, Research and Development, P.O. Box 5400, Princeton, New Jersey 08543-5400, United States

2. Departments of Discovery Chemistry, ⊥Biology, and #Preclinical Candidate Optimization, Biocon Bristol-Myers Squibb Research Center (BBRC), Bangalore 560099, India

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.6b00117

Reference20 articles.

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