Discovery of Novel PTP1B Inhibitors Derived from the BH3 Domain of Proapoptotic Bcl-2 Proteins with Antidiabetic Potency-Reference-Cited by-同舟云学术

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Discovery of Novel PTP1B Inhibitors Derived from the BH3 Domain of Proapoptotic Bcl-2 Proteins with Antidiabetic Potency

Published:2021-05-19 Issue:6 Volume:12 Page:1017-1023
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Zhang Chuanliang¹²³^ORCID,Wu Lijuan²³,Liu Xiaochun²³,Gao Jiangming²³,Liu Shan²³,Wu Juan²³,Huang Dingmin¹,Wang Zhenwei¹,Su Xianbin¹

Affiliation:

1. College of Chemical Engineering, Qingdao University of Science and Technology, Qingdao 266042, China

2. School of Medicine and Pharmacy, Ocean University of China, Qingdao 266003, China

3. Marine Biomedical Research Institute, Qingdao 266071, China

Funder

National Natural Science Foundation of China

Natural Science Foundation of Shandong Province

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.1c00174

Reference53 articles.

1. The Bcl2 family: regulators of the cellular life-or-death switch

2. The BCL-2 protein family, BH3-mimetics and cancer therapy

3. α/β-Peptide Foldamers Targeting Intracellular Protein–Protein Interactions with Activity in Living Cells

4. Evaluation of Diverse α/β-Backbone Patterns for Functional α-Helix Mimicry: Analogues of the Bim BH3 Domain

5. (α/β+α)-Peptide Antagonists of BH3 Domain/Bcl-xL Recognition: Toward General Strategies for Foldamer-Based Inhibition of Protein−Protein Interactions

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2. Biophysical Rationale for the Selective Inhibition of PTP1B over TCPTP by Nonpolar Terpenoids;The Journal of Physical Chemistry B;2023-09-20

3. Role of Protein Tyrosine Phosphatase 1B Inhibitor in Early Brain Injury of Subarachnoid Hemorrhage in Mice;Brain Sciences;2023-05-18

4. A biophysical rationale for the selective inhibition of PTP1B over TCPTP by nonpolar terpenoids;2023-04-18

5. Discovery of Novel PTP1B Inhibitors with Once-Weekly Therapeutic Potential for Type 2 Diabetes: Design, Synthesis, and In Vitro and In Vivo Investigations of BimBH3 Peptide Analogues;Journal of Medicinal Chemistry;2023-02-07

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