Development of Chimeric Molecules That Degrade the Estrogen Receptor Using Decoy Oligonucleotide Ligands

Author:

Naganuma Miyako123,Ohoka Nobumichi4,Tsuji Genichiro1ORCID,Tsujimura Haruna12,Matsuno Kenji3ORCID,Inoue Takao4,Naito Mikihiko5,Demizu Yosuke12ORCID

Affiliation:

1. Division of Organic Chemistry, National Institute of Health Sciences, Kanagawa 210-9501, Japan

2. Graduate School of Medical Life Science, Yokohama City University, Kanagawa 236-0027, Japan

3. Department of Chemistry and Life Science, Kogakuin University, Tokyo 192-0015, Japan

4. Division of Molecular Target and Gene Therapy Products, National Institute of Health Sciences, Kanagawa 158-8501, Japan

5. Laboratory of Targeted Protein Degradation, Graduate School of Pharmaceutical Sciences, The University of Tokyo, Tokyo 113-0033, Japan

Funder

Naito Foundation

Foundation for Promotion of Cancer Research

Takeda Science Foundation

Japan Foundation of Applied Enzymology

Sumitomo Foundation

Japan Agency for Medical Research and Development

Terumo Foundation for Life Sciences and Arts

Kobayashi Foundation for Cancer Research

NOVARTIS Foundation (Japan) for the Promotion of Science

Tokyo Biochemical Research Foundation

Japan Society for the Promotion of Science

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

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