Selective A<sub>3</sub> Adenosine Receptor Antagonist Radioligand for Human and Rodent Species-Reference-Cited by-同舟云学术

Selective A₃ Adenosine Receptor Antagonist Radioligand for Human and Rodent Species

Published:2022-03-02 Issue:4 Volume:13 Page:623-631
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Suresh R. Rama¹,Gao Zhan-Guo¹,Salmaso Veronica¹,Chen Eric¹,Campbell Ryan G.¹,Poe Russell B.²,Liston Theodore E.²,Jacobson Kenneth A.¹^ORCID

Affiliation:

1. Molecular Recognition Section, Laboratory of Bioorganic Chemistry, National Institute of Diabetes and Digestive and Kidney Diseases, Bethesda, Maryland 20892, United States

2. Astrocyte Pharmaceuticals, Cambridge, Massachusetts 02142, United States

Funder

National Institute of Diabetes and Digestive and Kidney Diseases

National Heart, Lung, and Blood Institute

National Institute of Mental Health

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.1c00685

Reference46 articles.

1. A3Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy

2. CF102 an A3 adenosine receptor agonist mediates anti-tumor and anti-inflammatory effects in the liver

3. The stimulation of A3 adenosine receptors reduces bone-residing breast cancer in a rat preclinical model

4. Suppressive roles of A3AR and TMIGD3 i1 in osteosarcoma malignancy

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