Cysteine-Targeted Insecticides against A. gambiae Acetylcholinesterase Are Neither Selective nor Reversible Inhibitors-Reference-Cited by-同舟云学术

Cysteine-Targeted Insecticides against A. gambiae Acetylcholinesterase Are Neither Selective nor Reversible Inhibitors

Published:2019-11-26 Issue:1 Volume:11 Page:65-71
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Gorecki Lukas¹²,Andrys Rudolf³,Schmidt Monika¹³,Kucera Tomas²,Psotka Miroslav¹³,Svobodova Barbora¹²,Hrabcova Veronika³²^ORCID,Hepnarova Vendula¹²,Bzonek Petr³²,Jun Daniel¹²,Kuca Kamil³^ORCID,Korabecny Jan¹²^ORCID,Musilek Kamil¹³⁴^ORCID

Affiliation:

1. University Hospital Hradec Kralove, Biomedical Research Centre, Sokolska 581, 500 05 Hradec Kralove, Czech Republic

2. University of Defence, Department of Toxicology and Military Pharmacy, Faculty of Military Health Sciences, Trebesska 1575, 500 01 Hradec Kralove, Czech Republic

3. University of Hradec Kralove, Faculty of Science, Department of Chemistry, Rokitanskeho 62, 500 03 Hradec Kralove, Czech Republic

4. Florida International University, Herbert Wertheim College of Medicine, Department of Cellular Biology & Pharmacology, 11200 SW Eighth Street GL 495-G Miami, Florida 33199, United States

Funder

Ministerstvo Zdravotnictví Ceské Republiky

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.9b00477

Reference27 articles.

1. World Malaria Report 2016; World Health Organization: Geneva; 2016. Licence: CC BY-NC-SA 3.0 IGO.

2. Inheritance of soybean aphid resistance in 21 soybean plant introductions

3. Insect Acetylcholinesterase as a Target for Effective and Environmentally Safe Insecticides