Systematically Mitigating the p38α Activity of Triazole-based BET Inhibitors
Author:
Affiliation:
1. Department of Chemistry, University of Minnesota Twin Cities, Minneapolis, Minnesota 55455, United States
Funder
American Cancer Society
University of Minnesota
National Institute of General Medical Sciences
Masonic Cancer Center, University of Minnesota
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Drug Discovery,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.9b00227
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1. The bromodomain interaction module
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4. Clinical trials for BET inhibitors run ahead of the science
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