Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition-Reference-Cited by-同舟云学术

Identification of the 2-Benzoxazol-2-yl-phenol Scaffold as New Hit for JMJD3 Inhibition

Published:2019-02-25 Issue:4 Volume:10 Page:601-605
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Giordano Assunta¹²,Forte Giovanni²,Terracciano Stefania²,Russo Alessandra²,Sala Marina²^ORCID,Scala Maria C.²,Johansson Catrine³,Oppermann Udo³,Riccio Raffaele²,Bruno Ines²,Di Micco Simone²^ORCID

Affiliation:

1. Institute of Biomolecular Chemistry (ICB), Consiglio Nazionale delle Ricerche (CNR), Via Campi Flegrei 34, I-80078 Pozzuoli, Napoli, Italy

2. Department of Pharmacy, University of Salerno, Via Giovanni Paolo II, 132, I-84084 Fisciano, Salerno, Italy

3. Botnar Research Centre, Oxford NIHR BRU, Oxford University, Oxford Centre for Translational Myeloma Research, Oxford, OX3 7LD, U.K.

Funder

Associazione Italiana per la Ricerca sul Cancro (AIRC) and Fondazione Cariplo

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.8b00589

Reference33 articles.

1. A selective jumonji H3K27 demethylase inhibitor modulates the proinflammatory macrophage response

2. Inhibitors of Protein Methyltransferases and Demethylases

3. Epigenetic drug discovery: a success story for cofactor interference

4. Utx Is Required for Proper Induction of Ectoderm and Mesoderm during Differentiation of Embryonic Stem Cells

5. The Histone H3 Lysine-27 Demethylase Jmjd3 Links Inflammation to Inhibition of Polycomb-Mediated Gene Silencing

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