N-Acylbenzenesulfonamide Dihydro-1,3,4-oxadiazole Hybrids: Seeking Selectivity toward Carbonic Anhydrase Isoforms-Reference-Cited by-同舟云学术

N-Acylbenzenesulfonamide Dihydro-1,3,4-oxadiazole Hybrids: Seeking Selectivity toward Carbonic Anhydrase Isoforms

Published:2017-07-02 Issue:8 Volume:8 Page:792-796
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Bianco Giulia¹,Meleddu Rita¹,Distinto Simona¹^ORCID,Cottiglia Filippo¹^ORCID,Gaspari Marco²^ORCID,Melis Claudia¹,Corona Angela¹,Angius Rossella³,Angeli Andrea⁴,Taverna Domenico²,Alcaro Stefano⁵,Leitans Janis⁶,Kazaks Andris⁶,Tars Kaspars⁶,Supuran Claudiu T.⁴^ORCID,Maccioni Elias¹

Affiliation:

1. Department of Life and Environmental Sciences, University of Cagliari, Via Ospedale 72, 09124 Cagliari, Italy

2. Department of Experimental and Clinical Medicine, “Magna Græcia” University of Catanzaro, 88100 Catanzaro, Italy

3. Laboratorio NMR e Tecnologie Bioanalitiche, Sardegna Ricerche, 09010 Pula (CA), Italy

4. Dipartimento NEUROFARBA, Sezione di Scienze Farmaceutiche, Università degli Studi di Firenze, Sesto Fiorentino, Florence, Italy

5. Dipartimento di Scienze della Salute, Università Magna Graecia di Catanzaro, Campus ‘S. Venuta’, Viale Europa, 88100 Catanzaro, Italy

6. Latvian Biomedical Research and Study Center, Ratsupites 1, Riga, Latvia

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

http://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.7b00205

Reference28 articles.

1. Entrapment of Carbon Dioxide in the Active Site of Carbonic Anhydrase II

2. Advances in structure-based drug discovery of carbonic anhydrase inhibitors

3. Carbonic Anhydrases An Overview

4. Carbonic anhydrase inhibitors: Valdecoxib binds to a different active site region of the human isoform II as compared to the structurally related cyclooxygenase II ‘selective’ inhibitor celecoxib

5. Effects of Brinzolamide, a Topical Carbonic Anhydrase Inhibitor, on Corneal Endothelial Cells

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