Design, Synthesis, and Evaluation of Tetrahydropyrrolo[1,2-c]pyrimidines as Capsid Assembly Inhibitors for HBV Treatment-Reference-Cited by-同舟云学术

Design, Synthesis, and Evaluation of Tetrahydropyrrolo[1,2-c]pyrimidines as Capsid Assembly Inhibitors for HBV Treatment

Published:2017-08-30 Issue:9 Volume:8 Page:969-974
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Li Xiaolin¹,Zhou Kai¹,He Haiying¹,Zhou Qiong¹,Sun Ya¹,Hou Lijuan¹,Shen Liang¹,Wang Xiaofei¹,Zhou Yuedong¹,Gong Zhen¹,He Shibo¹,Jin Huangtao¹,Gu Zhengxian¹,Zhao Shuyong²,Zhang Long²,Sun Chunyan²,Zheng Shansong²,Cheng Zhe²,Zhu Yidong²,Zhang Minghui²,Li Jian¹,Chen Shuhui¹

Affiliation:

1. WuXi AppTec (Shanghai) Co., Ltd., 288 FuTe Zhong Road, Shanghai 200131, P. R. China

2. Shandong Provincial Key Laboratory of Small Molecular Targeted Drugs, Qilu Pharmaceutical Co., Ltd., No. 243 Gong Ye Bei Road, Jinan, Shandong Province 250100, P. R. China

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.7b00288

Reference26 articles.

1. A new series of HAPs as anti-HBV agents targeting at capsid assembly

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