HTS by NMR for the Identification of Potent and Selective Inhibitors of Metalloenzymes-Reference-Cited by-同舟云学术

HTS by NMR for the Identification of Potent and Selective Inhibitors of Metalloenzymes

Published:2018-01-19 Issue:2 Volume:9 Page:137-142
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Baggio Carlo¹,Cerofolini Linda²,Fragai Marco²^ORCID,Luchinat Claudio²,Pellecchia Maurizio¹^ORCID

Affiliation:

1. Division of Biomedical Sciences, School of Medicine, University of California—Riverside, Riverside, California 92521, United States

2. Magnetic Resonance Center (CERM), University of Florence and Consorzio Interuniversitario Risonanze Magnetiche di Metallo Proteine (CIRMMP), Via L. Sacconi 6, 50019 Sesto Fiorentino, Italy

Funder

National Cancer Institute

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.7b00483

Reference40 articles.

1. NMR-Based Approaches for the Identification and Optimization of Inhibitors of Protein–Protein Interactions

2. Solution Nuclear Magnetic Resonance Spectroscopy Techniques for Probing Intermolecular Interactions

3. Perspectives on NMR in drug discovery: a technique comes of age

4. Discovery of Potent Nonpeptide Inhibitors of Stromelysin Using SAR by NMR

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