Discovery of New Selenoureido Analogues of 4-(4-Fluorophenylureido)benzenesulfonamide as Carbonic Anhydrase Inhibitors-Reference-Cited by-同舟云学术

Discovery of New Selenoureido Analogues of 4-(4-Fluorophenylureido)benzenesulfonamide as Carbonic Anhydrase Inhibitors

Published:2017-08-14 Issue:9 Volume:8 Page:963-968
ISSN:1948-5875
Container-title:ACS Medicinal Chemistry Letters
language:en
Short-container-title:ACS Med. Chem. Lett.

Author:

Angeli Andrea¹,Tanini Damiano²,Peat Thomas S.³,Di Cesare Mannelli Lorenzo⁴,Bartolucci Gianluca¹^ORCID,Capperucci Antonella²,Ghelardini Carla⁴,Supuran Claudiu T.¹^ORCID,Carta Fabrizio¹^ORCID

Affiliation:

1. University of Florence, NEUROFARBA Dept., Sezione di Scienze Farmaceutiche, Via Ugo Schiff 6, 50019 Sesto Fiorentino, Florence, Italy

2. University of Florence, Department of Chemistry “Ugo Schiff”, Via della Lastruccia 13, I-50019 Sesto Fiorentino, Florence, Italy

3. CSIRO, 343 Royal Parade, Parkville, Victoria 3052, Australia

4. NEUROFARBA Department, Section of Pharmacology and Toxicology, Università degli Studi di Firenze, Viale Pieraccini 6, 50139 Florence, Italy

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Drug Discovery,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acsmedchemlett.7b00280

Reference31 articles.

1. Bioisosterism: A Rational Approach in Drug Design

2. Bioisosterism: A Useful Strategy for Molecular Modification and Drug Design

3. Kinetic and X-ray crystallographic investigations on carbonic anhydrase isoforms I, II, IX and XII of a thioureido analog of SLC-0111

4. Safety Study of SLC-0111 in Subjects With Advanced Solid Tumours.https://clinicaltrials.gov/ct2/show/NCT02215850.

5. Targeting Tumor Hypoxia: Suppression of Breast Tumor Growth and Metastasis by Novel Carbonic Anhydrase IX Inhibitors

Cited by 60 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Iodine/Oxone® oxidative system for the synthesis of selenylindoles bearing a benzenesulfonamide moiety as carbonic anhydrase I, II, IX, and XII inhibitors;Organic & Biomolecular Chemistry;2024

2. Carbonic anhydrase inhibitor-decorated semiconducting oligomer nanoparticles for active-targeting NIR-II fluorescence tumor imaging;Nanotechnology;2023-09-11

3. A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation;Bioorganic & Medicinal Chemistry Letters;2023-09

4. 1,5-Diaryl-1,2,4-triazole Ureas as New SLC-0111 Analogues Endowed with Dual Carbonic Anhydrase and VEGFR-2 Inhibitory Activities;Journal of Medicinal Chemistry;2023-07-28

5. MM/GBSA prediction of relative binding affinities of carbonic anhydrase inhibitors: effect of atomic charges and comparison with Autodock4Zn;Journal of Computer-Aided Molecular Design;2023-03-17