An Aldol-Based Build/Couple/Pair Strategy for the Synthesis of Medium- and Large-Sized Rings: Discovery of Macrocyclic Histone Deacetylase Inhibitors-Reference-Cited by-同舟云学术

An Aldol-Based Build/Couple/Pair Strategy for the Synthesis of Medium- and Large-Sized Rings: Discovery of Macrocyclic Histone Deacetylase Inhibitors

Published:2010-11-10 Issue:47 Volume:132 Page:16962-16976
ISSN:0002-7863
Container-title:Journal of the American Chemical Society
language:en
Short-container-title:J. Am. Chem. Soc.

Author:

Marcaurelle Lisa A.¹,Comer Eamon¹,Dandapani Sivaraman¹,Duvall Jeremy R.¹,Gerard Baudouin¹,Kesavan Sarathy¹,Lee Maurice D.¹,Liu Haibo¹,Lowe Jason T.¹,Marie Jean-Charles¹,Mulrooney Carol A.¹,Pandya Bhaumik A.¹,Rowley Ann¹,Ryba Troy D.¹,Suh Byung-Chul¹,Wei Jingqiang¹,Young Damian W.¹,Akella Lakshmi B.¹,Ross Nathan T.¹,Zhang Yan-Ling¹,Fass Daniel M.¹,Reis Surya A.¹,Zhao Wen-Ning¹,Haggarty Stephen J.¹,Palmer Michelle¹,Foley Michael A.¹

Affiliation:

1. Chemical Biology Platform and Stanley Center for Psychiatric Research, Broad Institute of MIT and Harvard, 7 Cambridge Center, Cambridge, Massachusetts 02142, United States, and Center for Human Genetic Research, Massachusetts General Hospital, Harvard Medical School, Boston, Massachusetts 02114, United States

Publisher

American Chemical Society (ACS)

Subject

Colloid and Surface Chemistry,Biochemistry,General Chemistry,Catalysis

Link

https://pubs.acs.org/doi/pdf/10.1021/ja105119r

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