Development of a Large Scale Asymmetric Synthesis of the Glucocorticoid Agonist BI 653048 BS H3PO4-Reference-Cited by-同舟云学术

Development of a Large Scale Asymmetric Synthesis of the Glucocorticoid Agonist BI 653048 BS H3PO4

Published:2013-04-01 Issue:8 Volume:78 Page:3616-3635
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Reeves Jonathan T.¹,Fandrick Daniel R.¹,Tan Zhulin¹,Song Jinhua J.¹,Rodriguez Sonia¹,Qu Bo¹,Kim Soojin¹,Niemeier Oliver²,Li Zhibin¹,Byrne Denis¹,Campbell Scot³,Chitroda Ashish¹,DeCroos Phil¹,Fachinger Thomas²,Fuchs Victor¹,Gonnella Nina C.³,Grinberg Nelu¹,Haddad Nizar¹,Jäger Burkhard²,Lee Heewon¹,Lorenz Jon C.¹,Ma Shengli¹,Narayanan Bikshandarkoil A.¹,Nummy Larry J.¹,Premasiri Ajith¹,Roschangar Frank¹,Sarvestani Max¹,Shen Sherry¹,Spinelli Earl¹,Sun Xiufeng¹,Varsolona Richard J.¹,Yee Nathan¹,Brenner Michael²,Senanayake Chris H.¹

Affiliation:

1. Chemical Development, Boehringer Ingelheim Pharmaceuticals, Inc., 900 Old Ridgebury Road, P.O. Box 368, Ridgefield, Connecticut, 06877-0368, United States

2. Boehringer Ingelheim GmbH & Co. KG, Binger Strasse 173, 55216 Ingelheim am Rhein, Germany

3. Analytical Development, Boehringer Ingelheim Pharmaceuticals, Inc., 900 Old Ridgebury Road, P.O. Box 368, Ridgefield, Connecticut, 06877-0368, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo400079z

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