The Pthaladyns: GTP Competitive Inhibitors of Dynamin I and II GTPase Derived from Virtual Screening-Reference-Cited by-同舟云学术

The Pthaladyns: GTP Competitive Inhibitors of Dynamin I and II GTPase Derived from Virtual Screening

Published:2010-06-24 Issue:14 Volume:53 Page:5267-5280
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Odell Luke R.¹,Howan Dian¹,Gordon Christopher P.¹,Robertson Mark J.¹,Chau Ngoc²,Mariana Anna²,Whiting Ainslie E.²,Abagyan Ruben³,Daniel James A.²,Gorgani Nick N.²,Robinson Phillip J.²,McCluskey Adam¹

Affiliation:

1. Chemistry, The University of Newcastle, University Drive, Callaghan, NSW 2308, Australia

2. Cell Signaling Unit, Children's Medical Research Institute, The University of Sydney, 214 Hawkesbury Road, Westmead, NSW 2145, Australia

3. Department of Molecular Biology, The Scripps Research Institute, 10550 North Torrey Pines Road, TCP-28, La Jolla, California 92037

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm100442u

Reference57 articles.

1. Long chain amines and long chain ammonium salts as novel inhibitors of dynamin GTPase activity

2. Myristyl Trimethyl Ammonium Bromide and Octadecyl Trimethyl Ammonium Bromide Are Surface-Active Small Molecule Dynamin Inhibitors that Block Endocytosis Mediated by Dynamin I or Dynamin II

3. Small Molecule Inhibitors of Dynamin I GTPase Activity: Development of Dimeric Tyrphostins

4. Azido and Diazarinyl Analogues of Bis-Tyrphostin as Asymmetrical Inhibitors of Dynamin GTPase

5. From Spanish fly to room-temperature ionic liquids (RTILs): synthesis, thermal stability and inhibition of dynamin 1 GTPase by a novel class of RTILs

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