Lead Optimization of 17β-HSD1 Inhibitors of the (Hydroxyphenyl)naphthol Sulfonamide Type for the Treatment of Endometriosis-Reference-Cited by-同舟云学术

Lead Optimization of 17β-HSD1 Inhibitors of the (Hydroxyphenyl)naphthol Sulfonamide Type for the Treatment of Endometriosis

Published:2012-03-16 Issue:7 Volume:55 Page:3307-3318
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Henn Claudia¹²,Einspanier Almuth³,Marchais-Oberwinkler Sandrine¹,Frotscher Martin¹,Hartmann Rolf W.¹²

Affiliation:

1. Pharmaceutical and Medicinal Chemistry, Saarland University, Campus C2 3, D-66041 Saarbrücken, Germany

2. Helmholtz-Institute for Pharmaceutical Research Saarland (HIPS), Helmholtz Center for Infection Research (HZI), Campus C2 3, 66123 Saarbrücken, Germany

3. Faculty of Veterinary Medicine, Institute of Physiological Chemistry, An den Tierkliniken 1, 04103 Leipzig, Germany

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm201735j

Reference68 articles.

1. Involvement of up-regulation of 17?-hydroxysteroid dehydrogenase type 1 in maintenance of intratumoral high estradiol levels in postmenopausal breast cancers

2. 17Beta-hydroxysteroid dehydrogenase enzymes and breast cancer

3. Androgenic and estrogenic 17β-hydroxysteroid dehydrogenase/17-ketosteroid reductase in human ovarian epithelial tumors: evidence for the type 1, 2 and 5 isoforms

4. Disturbed estrogen and progesterone action in ovarian endometriosis

5. Endometriosis: Role of Ovarian Steroids in Initiation, Maintenance, and Suppression

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