The First Regioselective Palladium-Catalyzed Indolization of 2-Bromo- or 2-Chloroanilines with Internal Alkynes: A New Approach to 2,3-Disubstituted Indoles-Reference-Cited by-同舟云学术

The First Regioselective Palladium-Catalyzed Indolization of 2-Bromo- or 2-Chloroanilines with Internal Alkynes: A New Approach to 2,3-Disubstituted Indoles

Published:2004-10-01 Issue:22 Volume:6 Page:4129-4132
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Shen Ming¹,Li Guisheng¹,Lu Bruce Z.¹,Hossain Azad¹,Roschangar Frank¹,Farina Vittorio¹,Senanayake Chris H.¹

Affiliation:

1. Department of Chemical Development, Boehringer-Ingelheim Pharmaceuticals, Inc., 800 East Leigh Street, Suite 205, Richmond, Virginia 23219

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/ol048114t

Reference19 articles.

1. Marine natural products

2. Synthesis of indoles via palladium-catalyzed heteroannulation of internal alkynes

3. Synthesis of 2,3-Disubstituted Indoles via Palladium-Catalyzed Annulation of Internal Alkynes

4. Palladium-catalysed synthesis of heterocondensed pyrroles

Cited by 163 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. K₂CO₃-mediated annulation of 1,3-acetonedicarboxylates with 2-fluoro-1-nitroarenes: synthesis of indoles;Organic & Biomolecular Chemistry;2024

2. Divergent total syntheses of pyrroloiminoquinone alkaloids enabled by the development of a Larock/Buchwald–Hartwig annulation/cyclization;Chemical Science;2024

3. Electron Donor–Acceptor Complex Induced Fused Indoles with Hypervalent Iodine(III) Reagents;Organic Letters;2023-08-21

4. An Overview of Palladium-Catalyzed Fabrication of Some Heterocyclic Frameworks;Mini-Reviews in Organic Chemistry;2023-08

5. Quantitative analysis of steric effects on the regioselectivity of the Larock heteroannulation reaction;Organic & Biomolecular Chemistry;2023