Development of Orally Bioavailable Bicyclic Pyrazolones as Inhibitors of Tumor Necrosis Factor-α Production
Author:
Affiliation:
1. Health Care Research Center, Procter and Gamble Pharmaceuticals, 8700 Mason-Montgomery Road, Mason, Ohio 45040
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm049968m
Reference16 articles.
1. Recent reviews: (a) Adams, J. L.; Badger, A. M.; Kumar, S.; Lee, J. C. p38 MAP Kinase: Molecular target for the inhibition of pro-inflammatory cytokines.Progress in Medicinal Chemistry; King, F. D., Oxford, A. W., Eds.; Elsevier: Amsterdam, 2001; Vol. 38, pp 1−60. (b) Chen, Z.; Gibson, T. B.; Robinson, F.; Silvestro, L.; Pearson, G.; Xu, B.e.; Wright, A.; Vanderbilt, C.; Cobb, M. H. MAP Kinases.Chem. Rev.2001,101, 2449−2476.
2. Cytokines in autoimmunity
3. The Future Role of Anti-Tumour Necrosis Factor (TNF) Products in the Treatment of Rheumatoid Arthritis
4. 2,4,5- triarylimidazole inhibitors of IL-1 biosynthesis
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