The 1,4-Benzodiazepine-2,5-dione Small Molecule Template Results in Melanocortin Receptor Agonists with Nanomolar Potencies
Author:
Affiliation:
1. Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, Florida 32610
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm701303z
Reference70 articles.
1. Molecular cloning and expression of the human melanocyte stimulating hormone receptor cDNA
2. The Cloning of a Family of Genes That Encode the Melanocortin Receptors
3. The human melanocyte stimulating hormone receptor has evolved to become “super-sensitive” to melanocortin peptides
4. Identification of a receptor for gamma melanotropin and other proopiomelanocortin peptides in the hypothalamus and limbic system.
5. Molecular cloning of a novel melanocortin receptor.
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