Improving the Oral Efficacy of CNS Drug Candidates: Discovery of Highly Orally Efficacious Piperidinyl Piperidine M2 Muscarinic Receptor Antagonists
Author:
Affiliation:
1. Schering-Plough Research Institute, 2015 Galloping Hill Road, Kenilworth, New Jersey 07033
Publisher
American Chemical Society (ACS)
Subject
Drug Discovery,Molecular Medicine
Link
https://pubs.acs.org/doi/pdf/10.1021/jm0255163
Reference11 articles.
1. Experimental and computational approaches to estimate solubility and permeability in drug discovery and development settings
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