Benzopyrans Are Selective Estrogen Receptor β Agonists with Novel Activity in Models of Benign Prostatic Hyperplasia-Reference-Cited by-同舟云学术

Benzopyrans Are Selective Estrogen Receptor β Agonists with Novel Activity in Models of Benign Prostatic Hyperplasia

Published:2006-09-02 Issue:21 Volume:49 Page:6155-6157
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Norman Bryan H.¹,Dodge Jeffrey A.¹,Richardson Timothy I.¹,Borromeo Peter S.¹,Lugar Charles W.¹,Jones Scott A.¹,Chen Keyue¹,Wang Yong¹,Durst Gregory L.¹,Barr Robert J.¹,Montrose-Rafizadeh Chahrzad¹,Osborne Harold E.¹,Amos Robert M.¹,Guo Sherry¹,Boodhoo Amechand¹,Krishnan Venkatesh¹

Affiliation:

1. Discovery Chemistry Research, Bone and Inflammation Research, Lead Optimization Biology, Eli Lilly and Company, Lilly Corporate Center, Indianapolis, Indiana 46285

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm060491j

Reference18 articles.

1. Estrogen Receptor Modulators: Relationships of Ligand Structure, Receptor Affinity and Functional Activity

2. Discovery and Synthesis of [6-Hydroxy-3-[4-[2-(1-piperidinyl)ethoxy]phenoxy]- 2-(4-hydroxyphenyl)]benzo[b]thiophene: A Novel, Highly Potent, Selective Estrogen Receptor Modulator

3. Reflections on the Discovery and Significance of Estrogen Receptor β

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