Discovery and Synthesis of [6-Hydroxy-3-[4-[2-(1-piperidinyl)ethoxy]phenoxy]- 2-(4-hydroxyphenyl)]benzo[b]thiophene: A Novel, Highly Potent, Selective Estrogen Receptor Modulator-Reference-Cited by-同舟云学术

Discovery and Synthesis of [6-Hydroxy-3-[4-[2-(1-piperidinyl)ethoxy]phenoxy]- 2-(4-hydroxyphenyl)]benzo[b]thiophene: A Novel, Highly Potent, Selective Estrogen Receptor Modulator

Published:1997-05-01 Issue:10 Volume:40 Page:1407-1416
ISSN:0022-2623
Container-title:Journal of Medicinal Chemistry
language:en
Short-container-title:J. Med. Chem.

Author:

Palkowitz Alan D.¹,Glasebrook Andrew L.¹,Thrasher K. Jeff¹,Hauser Kenneth L.¹,Short Lorri L.¹,Phillips D. Lynn¹,Muehl Brian S.¹,Sato Masahiko¹,Shetler Pamela K.¹,Cullinan George J.¹,Pell Tina R.¹,Bryant Henry U.¹

Affiliation:

1. Lilly Research Laboratories, Eli Lilly and Company, Indianapolis, Indiana 46285

Publisher

American Chemical Society (ACS)

Subject

Drug Discovery,Molecular Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/jm970167b

Reference35 articles.

1. Raloxifene, tamoxifen, nafoxidine, or estrogen effects on reproductive and nonreproductive tissues in ovariectomized rats

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