Synthesis of 1-Hydroxy-Substituted Pyrazolo[3,4-c]- and Pyrazolo[4,3-c]quinolines and -isoquinolines from 4- and 5-Aryl-Substituted 1-Benzyloxypyrazoles-Reference-Cited by-同舟云学术

Synthesis of 1-Hydroxy-Substituted Pyrazolo[3,4-c]- and Pyrazolo[4,3-c]quinolines and -isoquinolines from 4- and 5-Aryl-Substituted 1-Benzyloxypyrazoles

Published:2000-12-01 Issue:26 Volume:65 Page:9001-9006
ISSN:0022-3263
Container-title:The Journal of Organic Chemistry
language:en
Short-container-title:J. Org. Chem.

Author:

Pawlas Jan¹,Vedsø Per¹,Jakobsen Palle¹,Huusfeldt Per Olaf¹,Begtrup Mikael¹

Affiliation:

1. Department of Medicinal Chemistry, The Royal Danish School of Pharmacy, Universitetsparken 2, DK-2100 Copenhagen, Denmark, and Novo Nordisk A/S, Medicinal Chemistry Research, Novo Nordisk Park, DK-2760 Måløv, Denmark

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/jo000986v

Reference16 articles.

1. Synthesis of 1,5-Diaryl-3-methyl-1 H-pyrazolo[4,5-c]isoquinolines and Studies of Binding to Specific Peripheral Benzodiazepine Binding Sites

2. Preparation of 5-Acyl- and 5-Aryl-Substituted 1-(Benzyloxy)pyrazoles via Directed Ortho-Lithiation/Transmetalation and Palladium Catalyzed Cross-Coupling

3. Synthesis of 4-Substituted 1-(Benzyloxy)pyrazoles via Iodine−Magnesium Exchange of 1-(Benzyloxy)-4-iodopyrazole

4. 1-Hydroxy-7-azabenzotriazole. An efficient peptide coupling additive

5. Selective carbon-carbon bond formation via transition metal catalysis. 3. A highly selective synthesis of unsymmetrical biaryls and diarylmethanes by the nickel- or palladium-catalyzed reaction of aryl- and benzylzinc derivatives with aryl halides

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