Enhancing activity and selectivity in a series of pyrrol-1-yl-1-hydroxypyrazole-based aldose reductase inhibitors: The case of trifluoroacetylation
Author:
Funder
VEGA
Aristotle University's Research Committee
Publisher
Elsevier BV
Subject
Organic Chemistry,Drug Discovery,Pharmacology,General Medicine
Reference43 articles.
1. Le mécanisme de la transformation de glucose en fructose par les vésicules séminales;Hers;Biochimica Biophysica Acta.,1956
2. Aldose reductase enzyme and its implication to major health problems of the 21(st) century;Alexiou;Curr. Med. Chem.,2009
3. From a dull enzyme to something else: facts and perspectives regarding aldose reductase;Del Corso;Curr. Med. Chem.,2008
4. Biochemistry and molecular cell biology of diabetic complications;Brownlee;Nature,2001
5. Oxidative stress and diabetic complications;Giacco;Circ. Res.,2010
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