Synthesis and Pharmacological Evaluation of [3H]HS665, a Novel, Highly Selective Radioligand for the Kappa Opioid Receptor-Reference-Cited by-同舟云学术

Synthesis and Pharmacological Evaluation of [3H]HS665, a Novel, Highly Selective Radioligand for the Kappa Opioid Receptor

Published:2014-12-24 Issue:3 Volume:6 Page:456-463
ISSN:1948-7193
Container-title:ACS Chemical Neuroscience
language:en
Short-container-title:ACS Chem. Neurosci.

Author:

Guerrieri Elena¹,Mallareddy Jayapal Reddy²,Tóth Géza²,Schmidhammer Helmut¹,Spetea Mariana¹

Affiliation:

1. Department of Pharmaceutical Chemistry, Institute of Pharmacy and Center for Molecular Biosciences (CMBI), University of Innsbruck, Innrain 80-82, A-6020 Innsbruck, Austria

2. Institute of Biochemistry, Biological Research Centre, Hungarian Academy of Sciences, Temesvari krt 62, H-6726 Szeged, Hungary

Publisher

American Chemical Society (ACS)

Subject

Cell Biology,Cognitive Neuroscience,Physiology,Biochemistry,General Medicine

Link

https://pubs.acs.org/doi/pdf/10.1021/cn5002792

Reference60 articles.

1. Challenges for opioid receptor nomenclature: IUPHAR Review 9

2. Peptide Kappa Opioid Receptor Ligands: Potential for Drug Development

3. Kappa opioids and the modulation of pain

4. Kappa Opioid Receptor Function

5. The dynorphin/κ-opioid receptor system and its role in psychiatric disorders

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