Expedient Synthesis of N-Methyl Tubulysin Analogues with High Cytotoxicity
Author:
Affiliation:
1. Department of Chemistry, University of California, Berkeley, California 94720
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/jo800384x
Reference51 articles.
1. Mechanism of Action of Tubulysin, an Antimitotic Peptide from Myxobacteria
2. Biological evaluation of tubulysin A: a potential anticancer and antiangiogenic natural product
3. Isolation, Crystal and Solution Structure Determination, and Biosynthesis of Tubulysins—Powerful Inhibitors of Tubulin Polymerization from Myxobacteria
4. Tubulysins, New Cytostatic Peptides from Myxobacteria Acting on Microtubuli. Production, Isolation, Physico-chemical and Biological Properties.
5. Total Synthesis of Tubulysin U and V
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