Canvass: A Crowd-Sourced, Natural-Product Screening Library for Exploring Biological Space

Author:

Kearney Sara E.1,Zahoránszky-Kőhalmi Gergely1,Brimacombe Kyle R.1,Henderson Mark J.1,Lynch Caitlin1,Zhao Tongan1,Wan Kanny K.12ORCID,Itkin Zina1,Dillon Christopher1,Shen Min1,Cheff Dorian M.1,Lee Tobie D.1,Bougie Danielle1,Cheng Ken1,Coussens Nathan P.1,Dorjsuren Dorjbal1,Eastman Richard T.1,Huang Ruili1,Iannotti Michael J.1,Karavadhi Surendra1,Klumpp-Thomas Carleen1,Roth Jacob S.1,Sakamuru Srilatha1,Sun Wei1,Titus Steven A.1,Yasgar Adam1,Zhang Ya-Qin1,Zhao Jinghua1,Andrade Rodrigo B.3ORCID,Brown M. Kevin4ORCID,Burns Noah Z.5ORCID,Cha Jin K.6ORCID,Mevers Emily E.7,Clardy Jon7ORCID,Clement Jason A.8,Crooks Peter A.9,Cuny Gregory D.10,Ganor Jake11,Moreno Jesus12,Morrill Lucas A.12,Picazo Elias12,Susick Robert B.12,Garg Neil K.12ORCID,Goess Brian C.13,Grossman Robert B.14ORCID,Hughes Chambers C.15ORCID,Johnston Jeffrey N.16ORCID,Joullie Madeleine M.17,Kinghorn A. Douglas18ORCID,Kingston David G.I.19ORCID,Krische Michael J.20,Kwon Ohyun12ORCID,Maimone Thomas J.21ORCID,Majumdar Susruta2223,Maloney Katherine N.24,Mohamed Enas25,Murphy Brian T.26ORCID,Nagorny Pavel27ORCID,Olson David E.282930ORCID,Overman Larry E.31ORCID,Brown Lauren E.32ORCID,Snyder John K.32,Porco John A.32ORCID,Rivas Fatima33,Ross Samir A.25ORCID,Sarpong Richmond34ORCID,Sharma Indrajeet35ORCID,Shaw Jared T.28ORCID,Xu Zhengren36,Shen Ben36ORCID,Shi Wei37ORCID,Stephenson Corey R.J.27ORCID,Verano Alyssa L.38,Tan Derek S.3839ORCID,Tang Yi12ORCID,Taylor Richard E.40,Thomson Regan J.41ORCID,Vosburg David A.2ORCID,Wu Jimmy42ORCID,Wuest William M.4344,Zakarian Armen45ORCID,Zhang Yufeng46,Ren Tianjing46,Zuo Zhong46ORCID,Inglese James1ORCID,Michael Sam1,Simeonov Anton1,Zheng Wei1,Shinn Paul1,Jadhav Ajit1,Boxer Matthew B.1,Hall Matthew D.1ORCID,Xia Menghang1,Guha Rajarshi1,Rohde Jason M.1ORCID

Affiliation:

1. National Center for Advancing Translational Sciences, National Institutes of Health, 9800 Medical Center Drive, Rockville, Maryland 20850, United States

2. Department of Chemistry, Harvey Mudd College, 301 Platt Boulevard, Claremont, California 91711, United States

3. Department of Chemistry, Temple University, 1901 North 13th Street, Philadelphia, Pennsylvania 19122, United States

4. Department of Chemistry, Indiana University, 800 East Kirkwood Avenue, Bloomington, Indiana 47405, United States

5. Department of Chemistry, Stanford University, 333 Campus Drive, Stanford, California 94305, United States

6. Department of Chemistry, Wayne State University, 5101 Cass Avenue, Detroit, Michigan 48202, United States

7. Department of Biological Chemistry and Molecular Pharmacology, Harvard Medical School, 240 Longwood Avenue, Boston, Massachusetts 02115, United States

8. Natural Products Discovery Institute, Baruch S. Blumberg Institute, 3805 Old Easton Road, Doylestown, Pennsylvania 18902, United States

9. University of Arkansas for Medical Sciences, 4301 West Markham Street 522, Little Rock, Arkansas 72205, United States

10. Department of Pharmacological and Pharmaceutical Sciences, University of Houston, 4849 Calhoun Road, Houston, Texas 77204, United States

11. Diamond Age Corp., 344 East Louisiana Street, McKinney, Texas 75069, United States

12. Department of Chemistry and Biochemistry, UCLA, 607 Charles E. Young Drive East, Los Angeles, California 90095, United States

13. Department of Chemistry, Furman University, 3300 Poinsett Highway, Greenville, South Carolina 29613, United States

14. Department of Chemistry, University of Kentucky, Lexington, Kentucky 40506, United States

15. Scripps Institution of Oceanography, UCSD, 9500 Gilman Drive, La Jolla, California 92093, United States

16. Department of Chemistry, Vanderbilt University, 7330 Stevenson Center, Nashville, Tennessee 37235, United States

17. Department of Chemistry, University of Pennsylvania, 231 South 34th Street, Philadelphia, Pennsylvania 19104, United States

18. College of Pharmacy, The Ohio State University, 500 West 12th Avenue, Columbus, Ohio 43210, United States

19. Department of Chemistry, Virginia Tech, 900 West Campus Drive, Blacksburg, Virginia 24061, United States

20. Chemistry Department, The University of Texas at Austin, 105 East 24th Street STOP A5300, Austin, Texas 78712, United States

21. Department of Chemistry, University of California Berkeley, 826 Latimer Hall, Berkeley, California 94720, United States

22. Department of Molecular Pharmacology and Neurology, Memorial Sloan Kettering Cancer Center, 1275 York Avenue, New York, New York 10065, United States

23. Center for Clinical Pharmacology, St Louis College of Pharmacy and Washington University School of Medicine, 2 Pharmacy Place, St. Louis, Missouri 63110, United States

24. Department of Chemistry, Point Loma Nazarene University, 3900 Lomaland Drive, San Diego, California 92106, United States

25. University of Mississippi School of Pharmacy, 2500 North State Street, Jackson, Mississippi 39216, United States

26. College of Pharmacy, Department of Medicinal Chemistry and Pharmacognosy, University of Illinois at Chicago, 900 South Ashland Avenue, Chicago, Illinois 60607, United States

27. Department of Chemistry, University of Michigan, 930 North University Avenue, Ann Arbor, Michigan 48109, United States

28. Department of Chemistry, University of California, Davis, One Shields Avenue, Davis, California 95616, United States

29. School of Medicine, Department of Biochemistry and Molecular Medicine, University of California, Davis, 2700 Stockton Boulevard, Suite 2102, Sacramento, California 95817, United States

30. Center for Neuroscience, University of California, Davis, 1544 Newton Court, Davis, California 95618, United States

31. Department of Chemistry, University of California, Irvine, Irvine, California 92697, United States

32. Department of Chemistry and Center for Molecular Discovery (BU-CMD), Boston University, 590 Commonwealth Avenue, Boston, Massachusetts 02215, United States

33. Department of Chemical Biology and Therapeutics, St. Jude Children’s Research Hospital, 262 Danny Thomas Place, Memphis, Tennessee 38105, United States

34. Department of Chemistry, University of California Berkeley, 841-A Latimer Hall, Berkeley, California 94720, United States

35. Department of Chemistry and Biochemistry, and Institute of Natural Products and Research Technologies, University of Oklahoma, 101 Stephenson Parkway, Norman, Oklahoma 73019, United States

36. Department of Chemistry, Florida Campus, The Scripps Research Institute, 130 Scripps Way, Jupiter, Florida 33458, United States

37. Department of Chemistry and Biochemistry, University of Arkansas, Fayetteville, Arkansas 72701, United States

38. Pharmacology Graduate Program, Weill Cornell Graduate School of Medical Sciences, Memorial Sloan Kettering Cancer Center, 1275 York Avenue, New York, New York 10065, United States

39. Chemical Biology Program, Sloan Kettering Institute and Tri-Institutional Research Program, Memorial Sloan Kettering Cancer Center, 1275 York Avenue, New York, New York 10065, United States

40. Department of Chemistry and Biochemistry and the Warren Family Research Center for Drug Discovery and Development, University of Notre Dame, 305 McCourtney Hall, Notre Dame, Indiana 46556, United States

41. Department of Chemistry, Northwestern University, 2145 Sheridan Road, Evanston, Illinois 60208, United States

42. Department of Chemistry, Dartmouth College, Hanover, New Hampshire 03755, United States

43. Department of Chemistry, Emory University, 1515 Dickey Drive, Atlanta, Georgia 30322, United States

44. Emory Antibiotic Resistance Center, Emory University School of Medicine, 201 Dowman Drive, Atlanta, Georgia 30322, United States

45. Santa Barbara Department of Chemistry and Biochemistry, University of California, Santa Barbara, California 93106, United States

46. School of Pharmacy, Faculty of Medicine, The Chinese University of Hong Kong, Sha Tin, New Territories, Hong Kong SAR

Funder

American Chemical Society

American Cancer Society

U.S. Department of Health and Human Services

National Science Foundation

Office of the Assistant Secretary of Defense for Health Affairs

Publisher

American Chemical Society (ACS)

Subject

General Chemical Engineering,General Chemistry

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