DCAF16-Based Covalent Handle for the Rational Design of Monovalent Degraders-Reference-Cited by-同舟云学术

DCAF16-Based Covalent Handle for the Rational Design of Monovalent Degraders

Published:2024-05-17 Issue:7 Volume:10 Page:1318-1331
ISSN:2374-7943
Container-title:ACS Central Science
language:en
Short-container-title:ACS Cent. Sci.

Author:

Lim Melissa¹²³,Cong Thang Do¹²³,Orr Lauren M.¹²³,Toriki Ethan S.¹²³,Kile Andrew C.²⁴,Papatzimas James W.²⁴^ORCID,Lee Elijah¹²³,Lin Yihan¹²³,Nomura Daniel K.¹²³⁵^ORCID

Affiliation:

1. Department of Chemistry, University of California, Berkeley, Berkeley, California 94720, United States

2. Novartis-Berkeley Translational Chemical Biology Institute, Berkeley, California 94720, United States

3. Innovative Genomics Institute, Berkeley, California 94720, United States

4. Novartis Biomedical Research, Emeryville, California 94608, United States

5. Department of Molecular and Cell Biology, University of California, Berkeley, Berkeley, California 94720, United States

Funder

Division of Chemistry

National Cancer Institute

Novartis Institutes for BioMedical Research

Mark Foundation For Cancer Research

Publisher

American Chemical Society (ACS)

Link

https://pubs.acs.org/doi/pdf/10.1021/acscentsci.4c00286

Reference37 articles.

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5. Chemoproteomics-enabled discovery of a covalent molecular glue degrader targeting NF-κB

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