Proximity-Induced Nucleic Acid Degrader (PINAD) Approach to Targeted RNA Degradation Using Small Molecules

Author:

Mikutis Sigitas1,Rebelo Maria2,Yankova Eliza34,Gu Muxin3,Tang Cong2,Coelho Ana R.2,Yang Mo5,Hazemi Madoka E.1,Pires de Miranda Marta2,Eleftheriou Maria34,Robertson Max1,Vassiliou George S.3,Adams David J.6,Simas J. Pedro27,Corzana Francisco8ORCID,Schneekloth John S.5,Tzelepis Konstantinos34ORCID,Bernardes Gonçalo J. L.12ORCID

Affiliation:

1. Yusuf Hamied Department of Chemistry, University of Cambridge, Lensfield Road, Cambridge CB2 1EW, U.K.

2. Instituto de Medicina Molecular João Lobo Antunes, Faculdade de Medicina, Universidade de Lisboa, Avenida Professor Egas Moniz, 1649-028, Lisboa, Portugal

3. Wellcome-MRC Cambridge Stem Cell Institute, University of Cambridge, Cambridge CB2 0AW, U.K.

4. Milner Therapeutics Institute, University of Cambridge, Puddicombe Way, Cambridge CB2 0AW, U.K.

5. Chemical Biology Laboratory, Center for Cancer Research, National Cancer Institute, Frederick, Maryland 21702, United States

6. Experimental Cancer Genetics, Wellcome Trust Sanger Institute, Hinxton, Cambridge CB10 1SA, U.K.

7. Católica Biomedical Research and Católica Medical School, Universidade Católica Portuguesa, 1649-023 Lisboa, Portugal

8. Departamento de Química, Centro de Investigación en Síntesis Química, Universidad de La Rioja, 26006 Logroño, Spain

Funder

Medical Research Council

Agencia Estatal de Investigaci?n

Leukaemia Foundation

Wellcome Trust

Cambridge Trust

Biotechnology and Biological Sciences Research Council

Cancer Research UK

Jardine Foundation

Publisher

American Chemical Society (ACS)

Subject

General Chemical Engineering,General Chemistry

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