Introduction of Trifluoroethylamine as Amide Isostere by C–H Functionalization of Heteroarenes
Author:
Affiliation:
1. Department of Discovery Chemistry, Genentech, Inc., 1 DNA Way, South San Francisco, California 94080, United States
2. Laboratoire de Synthèse Organique, UMR 7652 CNRS-École Polytechnique, Route de Saclay, 91128 Palaiseau Cedex, France
Publisher
American Chemical Society (ACS)
Subject
Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry
Link
https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.7b01880
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