Aerobic α,β-C(sp3)–H Bond Difunctionalization and C–N Bond Cleavage of Triethylamine: Difunctional Ammonium Iodide Enabling the Regioselective Synthesis of 4-Arylpyrimido[1,2-b]indazoles-Reference-Cited by-同舟云学术

Aerobic α,β-C(sp3)–H Bond Difunctionalization and C–N Bond Cleavage of Triethylamine: Difunctional Ammonium Iodide Enabling the Regioselective Synthesis of 4-Arylpyrimido[1,2-b]indazoles

Published:2019-07-18 Issue:15 Volume:21 Page:6074-6078
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Gao Qinghe¹^ORCID,Han Xinya²,Tong Peiyuan¹,Zhang Zhiang¹,Shen Haotian¹,Guo Yanrong²,Bai Suping¹

Affiliation:

1. School of Pharmacy, Xinxiang Medical University, Xinxiang, Henan 453003, P. R. China

2. School of Chemistry and Chemical Engineering, Anhui University of Technology, Maanshan, Anhui 243002, P. R. China

Funder

Ministry of Science and Technology of the People's Republic of China

National Natural Science Foundation of China

Anhui Province

Henan Province

State Key Laboratory of Microbial Technology, Shandong University

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.9b02218

Reference55 articles.

1. GdCl3 catalysed Grieco condensation: A facile approach for the synthesis of novel pyrimidine and annulated pyrimidine fused indazole derivatives in single pot under mild conditions and their anti-microbial activity

2. Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors

3. Synthetic Approaches to the New Drugs Approved During 2015

4. Synthesis and structure–activity relationships of novel pyrimido[1,2-b]indazoles as potential anticancer agents against A-549 cell lines

5. An approach towards the synthesis of novel fused nitrogen tricyclic heterocyclic scaffolds via GBB reaction

Cited by 38 articles. 订阅此论文施引文献订阅此论文施引文献，注册后可以免费订阅5篇论文的施引文献，订阅后可以查看论文全部施引文献

1. Synthesis, Characterization and Biological Evaluation of 3‐Oxo‐Pyrimido[1,2‐b]indazoles;Advanced Synthesis & Catalysis;2024-09-03

2. Cyclization Through Dual C(sp³)−H Functionalization;Advanced Synthesis & Catalysis;2024-08-22

3. Iodine Mediated Annulation of Triethylamine, Aldehydes and 2‐Aminopyridines for the Synthesis of 3‐Formyl‐Imidazo [1,2‐a]pyridine Derivatives;Advanced Synthesis & Catalysis;2024-08-14

4. I₂-DMSO-Mediated Construction of 2,3- and 2,4-Disubstituted Pyrimido[1,2-b]indazole Skeletons;The Journal of Organic Chemistry;2024-02-29

5. TBHP Mediated C–N Bond Cleavage of Tertiary Amines toward the Synthesis of Oxalamides and α,β-Epoxy Amides;The Journal of Organic Chemistry;2024-01-11