Fragment-Based Discovery of Pyrimido[1,2-<i>b</i>]indazole PDE10A Inhibitors-Reference-Cited by-同舟云学术

Fragment-Based Discovery of Pyrimido[1,2-b]indazole PDE10A Inhibitors

Published:2018 Issue:3 Volume:66 Page:286-294
ISSN:0009-2363
Container-title:Chemical and Pharmaceutical Bulletin
language:en
Short-container-title:CHEMICAL & PHARMACEUTICAL BULLETIN

Author:

Chino Ayaka¹,Seo Ryushi¹,Amano Yasushi¹,Namatame Ichiji¹,Hamaguchi Wataru¹,Honbou Kazuya¹,Mihara Takuma¹,Yamazaki Mayako¹,Tomishima Masaki¹,Masuda Naoyuki¹

Affiliation:

1. Drug Discovery Research, Astellas Pharma Inc.

Publisher

Pharmaceutical Society of Japan

Subject

Drug Discovery,General Chemistry,General Medicine

Link

https://www.jstage.jst.go.jp/article/cpb/66/3/66_c17-00836/_pdf

Reference36 articles.

1. 1) Rowley M., Bristow L. J., Hutson P. H., J. Med. Chem., 44, 477–501 (2001).

2. 2) Tandon R., Nasrallah H. A., Keshavan M. S., Schizophr. Res., 110, 1–23 (2009).

3. 3) Soderling S. H., Bayuga S. J., Beavo J. A., Proc. Natl. Acad. Sci. U.S.A., 96, 7071–7076 (1999).

4. 4) Loughney K., Snyder P. B., Uher L., Rosman G. J., Ferguson K., Florio V. A., Gene, 234, 109–117 (1999).

5. 5) Fujishige K., Kotera J., Michibata H., Yuasa K., Takebayashi S., Okumura K., Omori K., J. Biol. Chem., 274, 18438–18445 (1999).

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