Peptide to Peptoid Substitutions Increase Cell Permeability in Cyclic Hexapeptides-Reference-Cited by-同舟云学术

Peptide to Peptoid Substitutions Increase Cell Permeability in Cyclic Hexapeptides

Published:2015-06-05 Issue:12 Volume:17 Page:2928-2931
ISSN:1523-7060
Container-title:Organic Letters
language:en
Short-container-title:Org. Lett.

Author:

Schwochert Joshua¹,Turner Rushia¹,Thang Melissa¹,Berkeley Ray F¹,Ponkey Alexandra R¹,Rodriguez Kelsie M.¹,Leung Siegfried S F²,Khunte Bhagyashree³,Goetz Gilles³,Limberakis Chris³,Kalgutkar Amit S.⁴,Eng Heather⁵,Shapiro Michael J.³,Mathiowetz Alan M.⁶,Price David A.⁶,Liras Spiros⁶,Jacobson Matthew P.²,Lokey R. Scott¹

Affiliation:

1. Chemistry and Biochemistry University of California, Santa Cruz, California 95064, United States

2. Department of Pharmaceutical Chemistry, University of California, San Francisco, California 94158, United States

3. World Wide Medicinal Chemistry, Groton Laboratories, Pfizer Inc. Groton, Connecticut 06340, United States

4. Pharmacokinetics and Drug Metabolism, Cambridge Laboratories, Pfizer Inc. Cambridge, Massachusetts 02139, United States

5. Pharmacokinetics and Drug Metabolism, Groton Laboratories, Pfizer Inc. Groton, Connecticut 06340, United States

6. World Wide Medicinal Chemistry, Cambridge Laboratories, Pfizer Inc. Cambridge, Massachusetts 02139, United States

Publisher

American Chemical Society (ACS)

Subject

Organic Chemistry,Physical and Theoretical Chemistry,Biochemistry

Link

https://pubs.acs.org/doi/pdf/10.1021/acs.orglett.5b01162

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